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Review

Development of PARP inhibitors in oncology

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Pages 31-43 | Published online: 21 Nov 2008

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L. Schmidt, O. Sehic & C. Wild. (2022) Counting the cost of public and philanthropic R&D funding: the case of olaparib. Journal of Pharmaceutical Policy and Practice 15:1.
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Laurence Booth, Nichola Cruickshanks, Thomas Ridder, Yun Dai, Steven Grant & Paul Dent. (2013) PARP and CHK inhibitors interact to cause DNA damage and cell death in mammary carcinoma cells. Cancer Biology & Therapy 14:5, pages 458-465.
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Laura Orlando, Paola Schiavone, Palma Fedele, Nicola Calvani, Angelo Nacci, Margherita Cinefra, Maria D'Amico, Enrica Mazzoni, Antonella Marino, Francesco Sponziello, Franco Morelli, Lucia Lombardi, Nicola Silvestris & Saverio Cinieri. (2012) Poly (ADP-ribose) polymerase (PARP): rationale, preclinical and clinical evidences of its inhibition as breast cancer treatment. Expert Opinion on Therapeutic Targets 16:sup2, pages S83-S89.
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Nupur N. Gangopadhyay, James D. Luketich, Amy Opest, Carmen Visus, Ernest M. Meyer, Rodney Landreneau & Matthew J. Schuchert. (2011) Inhibition of Poly(ADP-Ribose) Polymerase (PARP) Induces Apoptosis in Lung Cancer Cell Lines. Cancer Investigation 29:9, pages 608-616.
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V Kruse, S Rottey, O De Backer, S Van Belle, V Cocquyt & H Denys. (2011) PARP INHIBITORS IN ONCOLOGY: A NEW SYNTHETIC LETHAL APPROACH TO CANCER THERAPY. Acta Clinica Belgica 66:1, pages 2-9.
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Carlos W. Nossa & Steven R. Blanke. (2010) Helicobacter pylori activation of PARP-1. Gut Microbes 1:6, pages 373-378.
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