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Review

The therapeutic potential of PDE4 inhibitors

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Pages 1301-1325 | Published online: 23 Feb 2005

Bibliography

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  • •Useful reference describing Pfizer's compound.
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  • •Useful reference describing Celltech's compound.
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  • •Useful reference describing RPR's compound.
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  • •Good review.
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  • •Useful reference describing SB's compound.
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  • T-440. Drugs of the future (1997) 22:729–732.
  • •Good review of Tanabe Seiyaku's compound.
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  • •Interesting paper detailing rabbit model.
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  • SOUNESS JE, RAO S: Proposal for pharmacologically distinct conformers of PDE4 cyclic AMP phosphodies-terases. Cell. Signal. (1997) 9(3/4):227–236.
  • •Interesting paper discussing the high and low affinity binding sites.
  • HUGHES B, OWENS R, PERRY M, WARRELLOW G, ALLEN R: PDE-4 inhibitors: the use of molecular-cloning in the design and development of novel drugs. Drug Discov. Today (1997) 2:89–101.
  • •Good review.
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  • •Good review.
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  • •Useful review.
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  • NORMAN P: PDE4 inhibitors 1998. Exp. Opin. Ther. Patents (1998) 8(7):771–784.
  • ••Excellent review.
  • BURNOUF C, PRUNIAUX M-P, SZILAGYI CM: Phosphodi-esterase 4 inhibitors. Ann. Reports. Med. Chem. (1998) 33:91–109.
  • ••Good review.
  • LAS-31025. Clin. Trials Monitor (1997) 69:25-26. Good review.
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  • ••Very useful review of Almirall's compound.
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  • ••Excellent review of SB's compound.
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  • •One of the few papers describing results of a clinical trial of a selective PDE4 inhibitor.
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  • Piclamilast. Drugs Future. (1998) 23:918–919.
  • •Useful review of RPR's compound.
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  • Analysts meeting (1998)
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