45
Views
0
CrossRef citations to date
0
Altmetric
Research Article

Effects of nano zinc oxide and nano chitosan on the taste masking paracetamol granules

& ORCID Icon
Received 03 Feb 2024, Accepted 03 May 2024, Published online: 21 May 2024

References

  • Nasr NEH, El Meshad AN, Fares AR. Nanocarrier systems in taste masking. Sci Pharm. 2022;90(1):20. doi: 10.3390/scipharm90010020.
  • Haser A, Zhang F. New strategies for improving the development and performance of amorphous solid dispersions. AAPS PharmSciTech. 2018;19(3):978–990. doi: 10.1208/s12249-018-0953-z.
  • Patil H, Tiwari RV, Repka MA. Hot-melt extrusion: from theory to application in pharmaceutical formulation. AAPS PharmSciTech. 2016;17(1):20–42. doi: 10.1208/s12249-015-0360-7.
  • Suzuki H, Onishi H, Hisamatsu S, et al. Acetaminophen-containing chewable tablets with suppressed bitterness and improved oral feeling. Int J Pharm. 2004;278(1):51–61. doi: 10.1016/j.ijpharm.2004.02.031.
  • Shelke M, Bidkar S, Dama G. A review: masking of taste unique approaches for bitter drug. World J Pharm Res. 2019;8(3):1429–1444. doi: 10.20959/wjpr20193-14415.
  • Kaushik P, Verma R, Mittal V, et al. Flavor microencapsulation for taste masking in medicated chewing gums—recent trends, challenges, and future perspectives. Coatings. 2022;12(11):1656. doi: 10.3390/coatings12111656.
  • Cram A, Breitkreutz J, Desset-Brèthes S, et al. Challenges of developing palatable oral paediatric formulations. Int J Pharm. 2009;365(1–2):1–3. doi: 10.1016/j.ijpharm.2008.09.015.
  • Chandrashekar J, Mueller KL, Hoon MA, et al. T2Rs function as bitter taste receptors. Cell. 2000;100(6):703–711. doi: 10.1016/S0092-8674(00)80706-0.
  • World Health Organization. Toolkit for research and development of paediatric antiretroviral drugs and formulations; 2018.
  • Hautala J, Heinämäki J, Hietala S, et al. Development of novel flavored Eudragit® E films for feline minitablet coatings. J Drug Delivery Sci Technol. 2016;34:41–50. doi: 10.1016/j.jddst.2016.03.003.
  • Simšič T, Nolimal B, Minova J, et al. A straw for paediatrics: how to administer highly dosed, bitter tasting paracetamol granules. Int J Pharm. 2021;602:120615. doi: 10.1016/j.ijpharm.2021.120615.
  • Banerjee S, Joshi U, Singh A, et al. Lipids for taste masking and taste assessment in pharmaceutical formulations. Chem Phys Lipids. 2021;235:105031. doi: 10.1016/j.chemphyslip.2020.105031.
  • Almurisi SH, Doolaanea AA, Akkawi ME, et al. Taste masking of paracetamol encapsulated in chitosan-coated alginate beads. J Drug Deliv Sci Technol. 2020;56:101520. doi: 10.1016/j.jddst.2020.101520.
  • Bladh N, Blychert E, Johansson K, et al. A new esomeprazole packet (sachet) formulation for suspension: in vitro characteristics and comparative pharmacokinetics versus intact capsules/tablets in healthy volunteers. Clin Ther. 2007;29(4):640–649. doi: 10.1016/j.clinthera.2007.03.014.
  • Wen H, Park K. Oral controlled release formulation design and drug delivery: theory to practice. Sussex, UK: John Wiley & Sons; 2011.
  • Al-Kasmi B, Alsirawan MB, Paradkar A, et al. Aqueous and pH dependent coacervation method for taste masking of paracetamol via amorphous solid dispersion formation. Sci Rep. 2021;11(1):8907. doi: 10.1038/s41598-021-88312-6.
  • Taki M, Tagami T, Ozeki T. Preparation of polymer-blended quinine nanocomposite particles by spray drying and assessment of their instrumental bitterness-masking effect using a taste sensor. Drug Dev Ind Pharm. 2017;43(5):715–722. doi: 10.1080/03639045.2016.1200070.
  • Nylese T, Rafaelsen J, Bolorizadeh M, et al. Streamlining identification of compounds in pharmaceutical drug products. Microsc Microanal. 2015;21(S3):553–554. doi: 10.1017/S1431927615003566.
  • Lee W, Shin TS, Ko S, et al. Control of dongchimi fermentation with chitosan deacetylated by alkali treatment to prevent over-ripening. J Food Sci. 2010;75(5):M308–M316. doi: 10.1111/j.1750-3841.2010.01643.x.
  • Younes I, Rinaudo M. Chitin and chitosan preparation from marine sources. Structure, properties and applications. Mar Drugs. 2015;13(3):1133–1174. doi: 10.3390/md13031133.
  • Mirzaei H, Darroudi M. Zinc oxide nanoparticles: biological synthesis and biomedical applications. Ceram Int. 2017;43(1):907–914. doi: 10.1016/j.ceramint.2016.10.051.
  • Bilensoy E, Varan C. Is there a niche for zinc oxide nanoparticles in future drug discovery? Expert Opin Drug Discov. 2023;18(9):943–945. doi: 10.1080/17460441.2023.2230152.
  • Pearnchob N, Siepmann J, Bodmeier R. Pharmaceutical applications of shellac: moisture-protective and taste-masking coatings and extended-release matrix tablets. Drug Dev Ind Pharm. 2003;29(8):925–938. doi: 10.1081/DDC-120024188.
  • Yajima T, Nogata A, Demachi M, et al. Particle design for taste-masking using a spray-congealing technique. Chem Pharm Bull. 1996;44(1):187–191. doi: 10.1248/cpb.44.187.
  • Shimano K, Kondo O, Miwa A, et al. Evaluation of uniform-sized microcapsules using a vibration-nozzle method. Drug Dev Ind Pharm. 1995;21(3):331–347. doi: 10.3109/03639049509048114.
  • Chukwu A, Agarwal S, Adikwu M. Some properties of chloroquine phosphate and quinine hydrochloride microcapsules. STP Pharma Sci. 1991;1(2):117–120.
  • Hashimoto Y, Tanaka M, Kishimoto H, et al. Preparation, characterization and taste-masking properties of polyvinylacetal diethylaminoacetate microspheres containing trimebutine. J Pharm Pharmacol. 2002;54(10):1323–1328. doi: 10.1211/002235702760345383.
  • Renu JD, Jalwal P, Singh B. Chewable tablets: a comprehensive review. Pharma Innov J. 2015;4(5):100–105.
  • Khandagade A, Kale V, Sinha R. Critical quality risk analysis of process parameters of fluid bed coating technology. IJIET. 2013;3:15–24.
  • Sangnim T, Huanbutta K. Development and evaluation of taste-masked paracetamol chewable tablets using a polymer and/or wax dispersion technique. J Drug Deliv Sci Technol. 2019;54:101361. doi: 10.1016/j.jddst.2019.101361.
  • Klang V, Valenta C, Matsko NB. Electron microscopy of pharmaceutical systems. Micron. 2013;44:45–74. doi: 10.1016/j.micron.2012.07.008.
  • Wilczyński S, Koprowski R, Duda P, et al. Microtomographic studies of subdivision of modified-release tablets. Int J Pharm. 2016;511(2):899–912. doi: 10.1016/j.ijpharm.2016.07.069.
  • Nylese T, Anderhalt R, Gorcea V. Identification of pharmaceutical constituents in finished product form using low kV microanalysis. Microsc Microanal. 2013;19(S2):272–273. doi: 10.1017/S1431927613003358.
  • Albertini B, Cavallari C, Passerini N, et al. Characterization and taste-masking evaluation of acetaminophen granules: comparison between different preparation methods in a high-shear mixer. Eur J Pharm Sci. 2004;21(2–3):295–303. doi: 10.1016/j.ejps.2003.10.017.
  • Shahoud S, Abdlwahed W, Hammad T. Development a taste-masked acetaminophen solid dispersions using Eudragit® E100 polymer by solvent evaporation technique. J Res Pharm. 2023;27(5):1998–2006. doi: 10.29228/jrp.479.
  • Shiino K, Iwao Y, Miyagishima A, et al. Optimization of a novel wax matrix system using aminoalkyl methacrylate copolymer E and ethylcellulose to suppress the bitter taste of acetaminophen. Int J Pharm. 2010;395(1–2):71–77. doi: 10.1016/j.ijpharm.2010.05.007.
  • Volić M, Pajić-Lijaković I, Djordjević V, et al. Alginate/soy protein system for essential oil encapsulation with intestinal delivery. Carbohydr Polym. 2018;200:15–24. doi: 10.1016/j.carbpol.2018.07.033.
  • Gryczke A, Schminke S, Maniruzzaman M, et al. Development and evaluation of orally disintegrating tablets (ODTs) containing ibuprofen granules prepared by hot melt extrusion. Colloids Surf B Biointerfaces. 2011;86(2):275–284. doi: 10.1016/j.colsurfb.2011.04.007.
  • Roblegg E, Dittrich P, Haltmeyer K, et al. Reformulation of a codeine phosphate liquid controlled-release product. Drug Dev Ind Pharm. 2010;36(12):1454–1462. doi: 10.3109/03639045.2010.487870.
  • Maniruzzaman M, Boateng JS, Bonnefille M, et al. Taste masking of paracetamol by hot-melt extrusion: an in vitro and in vivo evaluation. Eur J Pharm Biopharm. 2012;80(2):433–442. doi: 10.1016/j.ejpb.2011.10.019.
  • Gittings S, Turnbull N, Roberts CJ, et al. Dissolution methodology for taste masked oral dosage forms. J Control Release. 2014;173:32–42. doi: 10.1016/j.jconrel.2013.10.030.
  • Sarecka-Hujar B, Balwierz R, Ostrozka-Cieslik A, et al. Scanning electron microscopy and X-ray energy dispersive spectroscopy–useful tools in the analysis of pharmaceutical products. J Phys: conf Ser. 2017;931:012008. doi: 10.1088/1742-6596/931/1/012008.
  • Rodriguez L, Cavallari C, Passerini N, et al. Preparation and characterization by morphological analysis of diclofenac/PEG 4000 granules obtained using three different techniques. Int J Pharm. 2002;242(1–2):285–289. doi: 10.1016/S0378-5173(02)00189-8.
  • Klancke J. Dissolution testing of orally disintegrating tablets. Dissolution Technol. 2003;10(2):6–8. doi: 10.14227/DT100203P6.
  • Bilgili E, Rosen LA, Ko JS, et al. Experimental study of fluidized bed co-granulation of two active pharmaceutical ingredients: an industrial scale-up perspective. Part Sci Technol. 2011;29(3):285–309. doi: 10.1080/02726351.2010.516803.
  • To D, Davé RN. Fluid bed film coating of fine ibuprofen particles. Powder Technol. 2016;290:102–113. doi: 10.1016/j.powtec.2015.11.059.
  • Lid C-H, Chen S-C, Lee Y-C, et al. Directly compressible acetaminophen compositions prepared by fluidized-bed granulation. Drug Dev Ind Pharm. 1994;20(11):1911–1922. doi: 10.3109/03639049409050218.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.